Look up serotonergic in Wiktionary, the free dictionary. A serotonergic substance, medication, or receptor protein is one that affects neurotransmission...

the serotonin 5-HT2A receptor with serotonin, as well as with various serotonergic psychedelics, have been solved and published by Bryan L. Roth and colleagues...

consists of a group of symptoms that may occur with the use of certain serotonergic medications or drugs. The symptoms can range from mild to severe, and...

"expansion of consciousness". Also referred to as classic hallucinogens or serotonergic hallucinogens, the term psychedelic is sometimes used more broadly to...

transporter (NET). Inhibition of these transporters leads to an increase in serotonergic and noradrenergic signalling at postsynaptic receptors. Each drug blocks...

anxiety relief and sedation. Examples of trip killers, in the case of serotonergic psychedelics, include serotonin receptor antagonists, such as antipsychotics...

is a serotonin–norepinephrine–dopamine releasing agent (SNDRA) and serotonergic neurotoxin of the amphetamine family. It is used in scientific research...

A neuron (American English), neurone (British English), or nerve cell, is a cell that is excitable, firing electric signals called action potentials. Neurons...

striatal, hippocampal, prefrontal, and occipital serotonergic axon terminals. Neurotoxic damage to serotonergic axon terminals has been shown to persist for...

Noradrenergic and specific serotonergic antidepressants (NaSSAs) are a class of psychiatric drugs used primarily as antidepressants. They act by antagonizing...

receptor antagonist, is a drug used to inhibit the action of serotonin and serotonergic drugs at serotonin (5-HT) receptors. Antagonists of the 5-HT2A receptor...

4-Hydroxy-5-methoxytryptamine (4-HO-5-MeO-T) is a serotonergic neurotoxin of the tryptamine family. It is structurally related to the monoamine neurotransmitter...

This is a list of psychedelic drugs, also known as serotonergic psychedelics or classical hallucinogens. These drugs act specifically as serotonin 5-HT2A...

dopamine, and norepinephrine. Examples of monoamine neurotoxins include the serotonergic neurotoxins para-chloroamphetamine (PCA), methylenedioxymethamphetamine...

serotonin. The term was created to describe the mechanism of action of the serotonergic antidepressant vortioxetine, which acts as a serotonin reuptake inhibitor...

5-MAPB or MDAI, the stimulant 2-fluoromethamphetamine (2-FMA), and the serotonergic psychedelic 5-MeO-MiPT or 4-HO-MET, all at specific fixed doses. Contrary...

Monoaminergic activity enhancers (MAE), also known as catecholaminergic/serotonergic activity enhancers (CAE/SAE), are a class of drugs that enhance the action...

and paroxetine and consequently increased trazodone and mCPP levels. Serotonergic psychedelics like lysergic acid diethylamide (LSD) and psilocybin are...

4-methylenedioxyamphetamine (MDA) are well-known serotonergic neurotoxins that damage serotonergic neurons in the brain. However, MDMA and MDA injected...

perception disorder, possibly because both it and VSS involve changes in serotonergic synaptic transmission Drug-related visual snow, which can be caused by...

reduces serotonergic neuron firing. Over time, autoreceptor desensitization occurs, leading to increased serotonin release and enhanced serotonergic tone...

where the discriminative stimulus properties of LSD and presumably other serotonergic psychedelics in rats is mediated has been identified as the anterior...

and 5,7-dihydroxytryptamine (5,7-DHT). It is a relatively selective serotonergic neurotoxin, but also acts as a dopaminergic and noradrenergic neurotoxin...

mice and rats in association with serotonin 5-HT2A receptor activation. Serotonergic psychedelics like lysergic acid diethylamide (LSD) and psilocybin consistently...

Serotonin 5-HT2A receptor agonists can be divided into two main groups: (1) serotonergic psychedelics such as LSD, psilocybin, and mescaline; and (2) non-hallucinogenic...

also known as 6-OMe-DMT, is a serotonergic drug of the tryptamine family. It is the 6-methoxy derivative of the serotonergic psychedelic N,N-dimethyltryptamine...

is the largest serotonergic nucleus and provides a substantial proportion of the serotonin innervation to the forebrain. Serotonergic neurons are found...

Serotonergic cell groups refer to collections of neurons in the central nervous system that have been demonstrated by histochemical fluorescence to contain...

increased risk of serotonin syndrome when cyclobenzaprine was taken with the serotonergic drugs duloxetine or phenelzine. These substances may interact with cyclobenzaprine:...

4,5-Dihydroxytryptamine (4,5-DHT) is a serotonergic neurotoxin of the tryptamine family. It is structurally related to the monoamine neurotransmitter serotonin...

that the many serotonergic neurons innervate, these pathways are implicated in many functions, as listed above. The caudal serotonergic nuclei heavily...

as Lanmaoa asiatica. They may also sometimes be induced by classical serotonergic psychedelics such as mescaline and dimethyltryptamine (DMT), as well...

potential ergoline-based drugs include dopaminergic, antidopaminergic, serotonergic, and antiserotonergic. Ergoline alkaloids often interfere with multiple...

4-methylenedioxyamphetamine (MDA) are well-known serotonergic neurotoxins that damage serotonergic neurons in the brain. However, MDMA and MDA injected...

entactogen-like effects, such as the phenethylamine serotonergic psychedelic 2C-B and the atypical tryptamine serotonergic psychedelics 5-MeO-DiPT and 5-MeO-MiPT....

aggression. Known drugs with antiaggressive effects include various serotonergic agents, antidopaminergic drugs like antipsychotics, anticonvulsants and...

numerous projections from the mRN and dRN to key brain structures make serotonergic system fundamental in regulating brain homeostasis. However, studies...

4-methylenedioxy-N-methylamphetamine (MDMA) may not themselves be responsible for their serotonergic neurotoxicity, as an intracerebroventricular injection does not appear...

drugs, although targeted at dopaminergic receptors, cross-react with serotonergic 5-HT2B receptors as well, and have been reported to cause cardiac fibrosis...

is an American medicinal chemist known for his work in the areas of serotonergic and dopaminergic drugs as well as drug discrimination. He is most well...

psychedelic drug, a synthetic analogue of psilocybin, which has high serotonergic activity. It produces the head-twitch response, a behavioral proxy of...

(2,4-DCA) is a psychostimulant of the amphetamine family and a potent serotonergic neurotoxin related to para-chloroamphetamine (PCA; 4-chloroamphetamine)...

thus complements the classical serotonergic-opioid peptide descending pain-inhibiting system: whereas the serotonergic-opioid peptide pathway ultimately...

[citation needed] However, one proposed mechanism is the stimulation of serotonergic 5-HT receptors, particularly those involved in tactile sensation and...

9-methoxyibogaminalog, is a non-selective serotonin receptor modulator, serotonergic psychedelic, and psychoplastogen of the ibogalog group related to the...

Efavirenz (Sustiva) – has serotonergic psychedelic effects at supratherapeutic doses Ergonovine (ergometrine; Ergotrate) – has serotonergic psychedelic effects...

3-(2-piperidinoethyl)indole, is a serotonin receptor modulator and possible serotonergic psychedelic of the tryptamine family. It is the derivative of tryptamine...

4-methylenedioxyamphetamine (MDA) are well-known serotonergic neurotoxins that damage serotonergic neurons in the brain. However, MDMA and MDA injected...

anesthetics. Antipsychotics, which are dopamine receptor antagonists, and many serotonergic agents, such as meta-chlorophenylpiperazine (mCPP), can also produce...

function of pathways implicated with stress brains and anxiety, such as the serotonergic or GABAergic pathways. Though nicotine is typically associated with a...

para-Chlorophenethylamine (pCPE) also known as 4-chlorophenylethylamine, is a potent serotonergic drug that is a structural analog of para-chloroamphetamine, lacking a...

has been anecdotally reported to be a mild anaphrodisiac, as has the serotonergic empathogen MDMA, popularly known as "ecstasy". However, systematic study...

derivative and formerly as CYB005, is a serotonin receptor agonist and serotonergic psychedelic which is under development for use at non-hallucinogenic...

as 4-iodoamphetamine (4-IA), is a monoamine releasing agent (MRA) and serotonergic neurotoxin of the amphetamine family related to para-chloroamphetamine...

receptor was initially noted for its central role as the primary target of serotonergic psychedelic drugs such as LSD and psilocybin mushrooms. It later regained...

Mirtazapine has been used as a hallucinogen antidote to block the effects of serotonergic psychedelics like psilocybin and lysergic acid diethylamide (LSD). Mirtazapine...

Serotonin itself is too hydrophilic to enter serotonergic neurons without the SERT, whereas serotonergic psychedelics and serotonin's N-methylated metabolites...

Nonproprietary Name; developmental code name EMD-49980) is a dopaminergic and serotonergic drug which was under development for the treatment of major depressive...

function as antiemetics, however the clinical significance of this anti-serotonergic activity of memantine in Alzheimer's disease is unknown. Memantine acts...

receptor. The drug's route of administration has not been specified. Serotonergic psychedelics like psilocybin and lysergic acid diethylamide (LSD) are...

November 2022. Retrieved 16 February 2025. LSR 3000 is a small molecule, serotonergic neuroplasogen therapeutic being developed by Lusaris Therapeutics, for...

blocking the serotonin release and effects of MDMA, SSRIs fully block the serotonergic neurotoxicity of MDMA in animals. However, delayed administration of...

motivation. This syndrome may be related to serotonergic effects on the frontal lobes and/or serotonergic modulation of mid-brain dopaminergic systems...

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microdosing is a form of drug microdosing in which sub-hallucinogenic doses of serotonergic psychedelics like LSD and psilocybin are taken for claimed cognitive...

agonists as drugs are limited by their mediation of allergy-type symptoms. Serotonergic psychedelics, acting as serotonin 5-HT2A receptor agonists, such as LSD...

A close analogue of αMT, α-ethyltryptamine (αET), is known to be a serotonergic neurotoxin similarly to MDMA and para-chloroamphetamine (PCA). 2-Oxo-αMT...

simplified lysergamide which is closely related to the highly potent serotonergic psychedelic lysergic acid diethylamide (LSD). It is the analogue of LSD...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

dependence, was correlated with low basal dopaminergic activity, high serotonergic activity, and low basal noradrenergic activity, respectively. Many studies...

mushrooms (which contain the serotonin 5-HT2A receptor agonist and serotonergic psychedelic psilocybin) and Amanita muscaria mushrooms (which contain...

contributor of serotonergic agents, especially 5-HT to the hippocampus. These findings, together with the demonstration that serotonergic agents block long-term...

Receptor/signaling modulators • Adrenergics • Dopaminergics • Melatonergics • Serotonergics • Monoamine reuptake inhibitors • Monoamine releasing agents • Monoamine...

the thalamus/hypothalamus and a number of dopaminergic, noradrenergic, serotonergic, histaminergic, cholinergic, and glutamatergic brain nuclei. The ARAS...

Fenfluramine, sold under the brand name Fintepla, is a serotonergic medication used for the treatment of seizures associated with Dravet syndrome and Lennox–Gastaut...

Dimethyltryptamine (DMT), also known as N,N-dimethyltryptamine (N,N-DMT), is a serotonergic hallucinogen and investigational drug of the tryptamine family that occurs...

antidepressant with additional anxiolytic properties acting via dopaminergic and serotonergic mechanisms which was formerly marketed in France and Spain, as well as...

efavirenz, glaucine, IHCH-7113, MK-212, quipazine, RH-34) For a full list of serotonergic psychedelics, see the navbox here and the list here instead. Dissociatives...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

N-diallyltryptamine or as daltocin, is a serotonin receptor agonist and serotonergic psychedelic of the tryptamine and 4-hydroxytryptamine families. It has...

and simplified or partial ergoline that is structurally related to the serotonergic psychedelic lysergic acid diethylamide (LSD). It is the analogue of LSD...

albeit modestly, for apathy in dementia and Parkinson's disease. The DOx serotonergic psychedelic 2,5-dimethoxy-4-propylamphetamine (DOPR), which acts as an...

4-glutaryloxy-N,N-dimethyltryptamine (4-HO-DMT O-glutarate or 4-GO-DMT) is a serotonergic psychedelic of the tryptamine family. It acts as a prodrug of psilocin...

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DOPEGAL DSP-4 MDA (tenamfetamine) Oxidopamine (6-OHDA) Xylamine V-61 Serotonergic 2′-NH2-MPTP (2′-amino-MPTP) 2,4-DCA 2,4,5-THA 2,4,5-THMA pCPE 3-CA 3...

5-methoxytryptamine families. It has unique and distinct effects from other serotonergic tryptamines, including some stimulant- and entactogen-like effects, robust...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

setiptiline are also sometimes described as noradrenergic and specific serotonergic antidepressants (NaSSAs). Monoamine oxidase inhibitors include Isocarboxazid...

meta-chloroamphetamine (MCA), is a psychostimulant of the amphetamine family and a serotonergic neurotoxin related to para-chloroamphetamine (PCA; 4-chloroamphetamine)...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

the "Mount Everest of psychedelics". 5-MeO-DMT differs from most other serotonergic psychedelics in having much greater activity at the serotonin 5-HT1A...

Zolmitriptan, sold under the brand name Zomig among others, is a serotonergic medication which is used in the acute treatment of migraine attacks with...

5-dimethoxyphenethylamine, is a serotonin receptor modulator and possible serotonergic psychedelic of the phenethylamine and 2C families. 2C-CN was previously...

Fibromyalgia is potentially associated with polymorphisms of genes in the serotonergic, dopaminergic and catecholaminergic systems. Several genes have been...

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characterizes the development and function of unique populations of serotonergic neurons in the mouse brain. To enable this functional dissection, Dymecki...

N-Trimethylene-2C-TFM Drug class Selective serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen; Antidepressant ATC code None Legal status...

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patients have seen a lack of improvement from the use of antidepressants, serotonergic hallucinogens have been observed to be rather effective in treatment...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

(formerly Bufo alvarius, now Incilius alvarius), which contains the serotonergic psychedelic 5-MeO-DMT, and administer the venom to produce hallucinogenic...

MPTP is a selective dopaminergic neurotoxin, 2′-NH2-MPTP is a specific serotonergic and noradrenergic neurotoxin that does not affect dopaminergic neurons...

against serotonergic psychedelics or as a so-called "trip killer". The drug has been clinically studied in combination with the serotonergic psychedelic...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

genes with important neuronal implications, such as the BDNF gene and serotonergic genes. The brain-derived neurotrophic factor (BDNF) gene plays a role...

serotonin 5-HT2A receptor agonist and 2-benzylpiperidine analogue of the serotonergic psychedelic 25B-NBOMe which is used in scientific research. The (S,S)-isomer...

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neurotoxic to human midbrain dopaminergic neurons and, to a lesser extent, serotonergic neurons. Methamphetamine neurotoxicity causes adverse changes in brain...

releasing agent, a non-selective serotonin receptor agonist, and a serotonergic psychedelic. However, αMT levels are much lower than those of αMS with...

found in more than 200 species of mushrooms, with hallucinogenic and serotonergic effects. Effects include euphoria, changes in perception, a distorted...

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Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Drug class Serotonin 5-HT2A receptor agonist; Possible serotonergic psychedelic or hallucinogen ATC code None Identifiers IUPAC name...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

a boxed warning, that stated use of ondansetron in conjunction with serotonergic drugs (SSRIs, SNRIs, MAOIs and TCAs) had been linked to rare cases of...

5-methoxy-N-methyl-N-ethyltryptamine, is a serotonin receptor modulator, putative serotonergic psychedelic, and relatively rare designer drug of the tryptamine family...

4-dihydroxyamphetamine (HHA; α-methyldopamine), HHMA may be involved in the serotonergic neurotoxicity of MDMA. However, findings in this regard are conflicting...

tachycardia, hyperthermia, and serotonergic crisis, particularly in combination with monoamine oxidase inhibitors or other serotonergic substances. A meta-analysis...

in which it fully substitutes for, and additionally lacks any kind of serotonergic neurotoxicity. Hence, MDAT is considered likely to be a non-neurotoxic...

Relaxed Beliefs Under pSychedelics, is a model of affect concerning serotonergic psychedelics, associated with the theories of Karl Friston and Robin...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

acid amide (iso-LSA or iso-LA-819), isolysergamide, or erginine, is a serotonergic psychedelic of the ergoline and lysergamide families related to ergine...

extends to other serotonergic agents, including triptans, other tricyclic antidepressants, and tramadol. Fluvoxamine increases the serotonergic effects of clomipramine...

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α-methyl-5-hydroxytryptophan are prodrugs of α-methylserotonin that have serotonergic actions and have been suggested for potential therapeutic use. However...

Non-selective serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen Identifiers IUPAC name...

Other names MYCO004 Routes of administration Transdermal (patch) Drug class Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen...

of levodopa-derived dopamine release in the striatum is performed by serotonergic neurons that have no negative feedback mechanisms (they lack D2R receptors...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

N-diisopropyltryptamine; O-Propionyl-4-HO-DiPT Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

psychedelics, show distinct and dissimilar subjective effects from those of serotonergic psychedelics like LSD, psilocybin, and mescaline. Ibogaine and noribogaine...

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β-carbolines are said to be qualitatively distinct from and unlike those of serotonergic psychedelics like LSD but similar to those of ibogaine. Taken orally...

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vesicular monoamine transporter 2 (VMAT2) than MDMA and may have less serotonergic neurotoxicity. In contrast to certain other entactogens like MDMA, methylone...

Receptor/signaling modulators • Monoamine releasing agents • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

sensitivity, the so-called "gluten psychosis". It has been reported that in serotonergic hallucinations, the person maintains an awareness that they are hallucinating...

modulator of the tryptamine family. It is the 7-methoxy derivative of the serotonergic psychedelic dimethyltryptamine (DMT) and is a positional isomer of 5-MeO-DMT...

MSP-1014 is a serotonergic psychedelic which is under development for the treatment of major depressive disorder, other depressive disorders, and anxiety...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

the effects are more likely to resemble those of deliriants than of serotonergic psychedelics such as LSD. In 2006, two men who apparently ate the fish...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

activity is compatible with the definition of a noradrenergic and specific serotonergic antidepressant (NaSSA), and as such, S32212 could in turn be classified...

endocannabinoid neurotransmitters". As with terms such as dopaminergic and serotonergic, related proteins and cellular components involved in endocannabinoid...

interactions with tyramine-containing foods and some sympathomimetic or serotonergic drugs. Nevertheless, modern reviews and prescribing guides state that...

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TFMBOX is a putative serotonergic psychedelic of the phenethylamine and benzoxepin ("BOX") families. It is the cyclized phenethylamine analogue of DOTFM...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

inhibition. Serotonergic activity among phenidates is very rare, and 3,4-DCMP is one of only three compounds from this class with appreciable serotonergic activity...

4-methoxyamphetamine (4-MA), is a designer drug of the amphetamine class with serotonergic effects. Unlike other similar drugs of this family, PMA does not produce...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

v t e Antimigraine preparations (N02C) Analgesic/abortive Serotonergics Ergolines Dihydroergocryptine Dihydroergotamine Ergotamine (+caffeine, +chlorcyclizine/caffeine)...

as hallucinogen antidotes or "trip killers" to block the effects of serotonergic psychedelics like psilocybin and lysergic acid diethylamide (LSD). Among...

5-dimethoxy-N-(2-methoxybenzyl)amphetamine Drug class Serotonin 5-HT2 receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name 1-(2...

N-(2-Methoxybenzyl)-5-methoxytryptamine Drug class Serotonin 5-HT2 receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

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Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

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found in vertebrates. In humans, TPH2 is primarily expressed in the serotonergic neurons of the brain, with the highest expression in the raphe nucleus...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

have been determined to be dependent on the dopaminergic and possibly serotonergic neurotransmitter systems, its exact mechanism of action is unknown, and...

Receptor/signaling modulators • Adrenergics • Dopaminergics • Melatonergics • Serotonergics • Monoamine reuptake inhibitors • Monoamine releasing agents • Monoamine...

PolkaDot and Tre House. Both psilocybin and 4-AcO-DMT are prodrugs of the serotonergic psychedelic psilocin. Psychedelic mushroom stores operate in a legal...

N-diethyltryptamine; Ethacetin; Ethylacybin Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status DE:...

A potential risk of frequent repeated long-term use of LSD and other serotonergic psychedelics is cardiac fibrosis and valvulopathy due to serotonin 5-HT2B...

term "neuro" refers to the dense core granules, similar to those in serotonergic neurons that store monoamines. The term "endocrine" refers to the synthesis...

non-selective serotonin receptor agonist, serotonin 5-HT2A receptor agonist, serotonergic psychedelic – mental disorders [7] ALM-007 (ALM007) – undefined mechanism...

shows reduced psychostimulant-like effects, addictive potential, and serotonergic neurotoxicity. In clinical studies, (R)-MDMA produces similar effects...

results, including evidence pointing towards basal hyperactivity of serotonergic systems. Serotonin receptor and transporter binding studies have yielded...

N-(2-methoxybenzyl)-4-isopropylthio-2,5-dimethoxyphenethylamine, is a serotonergic psychedelic of the 25-NB (NBOMe) family. It is the NBOMe analogue of...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

1-Benzoyl-N,N-dimethyltryptamine; 1Bz-DMT; "Example 2-17" Drug class Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

Receptor/signaling modulators • Adrenergics • Dopaminergics • Melatonergics • Serotonergics • Monoamine reuptake inhibitors • Monoamine releasing agents • Monoamine...

v t e Antimigraine preparations (N02C) Analgesic/abortive Serotonergics Ergolines Dihydroergocryptine Dihydroergotamine Ergotamine (+caffeine, +chlorcyclizine/caffeine)...

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Non-selective serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

Histaminergic Melatonergic Monoaminergic Neurotransmission Opioidergic Serotonergic Froestl, Wolfgang (2011). "An historical perspective on GABAergic drugs"...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Non-selective serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

Drug class Serotonin 5-HT2A receptor partial agonist; Possible serotonergic psychedelic or hallucinogen ATC code None Identifiers IUPAC name 1-(4-bromo-2...

5-trimethoxyphenethylamine Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name 2-(2,6-dichloro-3...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

5-methylenedioxyphenethylamine Drug class Serotonin 5-HT2 receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

N-dimethyltryptamine Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name 1,1,2...

Routes of administration Oral Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

10-didehydroergolin-8β-yl)methanone Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name (2...

class Serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Receptor/signaling modulators • Monoamine releasing agents • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

derivative and putative serotonergic psychedelic. It is the O-acetylated analogue of the naturally occurring peripherally selective serotonergic tryptamine bufotenine...

Scale (HRS), are considerably less intense than those of conventional serotonergic psychedelics like psilocybin and dimethyltryptamine (DMT), and are more...

10-didehydroergoline-8-carboxamide; SYN-L-234 Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Identifiers CAS Number 3029080-72-3...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

N-dimethyltryptamine; 1A-5-MeO-DMT; 1-Ac-5-MeO-DMT; "Example 2-16" Drug class Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

2C-E-FLY Clinical data Drug class Serotonergic psychedelic; Hallucinogen Legal status Legal status In general unscheduled Identifiers IUPAC name 2-(8-Ethyl-2...

disorders. This would demonstrate little to zero cross-tolerance with serotonergic or lithium treatment. These drugs mimic three classes of endorphins,...

is also a potent serotonin 5-HT2A receptor agonist and hence may be a serotonergic psychedelic. The drug has been investigated in animals as a potential...

4-Methylthio-N,N-dimethyltryptamine Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name N...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name 2-[3-(difluoromethoxy)-4...

yclopropyltryptamine, is a psychedelic tryptamine derivative. It has serotonergic effects, and has reportedly been sold as a designer drug since around...

been found to possess antidepressant properties, mediated through the serotonergic and noradrenergic systems (although the precise mechanism remains to...

mianserin has sometimes been described as a noradrenergic and specific serotonergic antidepressant (NaSSA). However, the actual evidence in support of this...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Specifically, this side effect has been particularly associated with serotonergic antidepressants like SSRIs and SNRIs and may be less with atypical antidepressants...

DOPEGAL DSP-4 MDA (tenamfetamine) Oxidopamine (6-OHDA) Xylamine V-61 Serotonergic 2′-NH2-MPTP (2′-amino-MPTP) 2,4-DCA 2,4,5-THA 2,4,5-THMA pCPE 3-CA 3...

Oral, intramuscular injection Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status DE:...

from the enterochromaffin cells. B. dentium is able to modulate the serotonergic system in the brain as well as the intestine. In mice, colonisation of...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

pharmacological profile similar to that of LSD, acting primarily as a serotonergic hallucinogen. Analogues of 1S-LSD include 1P-LSD, 1D-LSD, 1T-LSD, 1V-LSD...

Chlorpromazine Serotonin syndrome; excessive serotonergic activity due usually to combined use of serotonergic drugs (e.g. antidepressants, stimulants, triptans)...

(DOIB or DOiBu) is a serotonin 5-HT2A receptor agonist, serotonergic psychedelic, and anti-inflammatory drug of the phenethylamine, amphetamine...

MMM; β-Aminodihydroasarone Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status US:...

for Emergencies. He is associated with REBUS, a neurological model of serotonergic psychedelics. In 1996, Friston received the first Young Investigators...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

Chlorphentermine, sold under the brand names Apsedon, Desopimon, and Lucofen, is a serotonergic appetite suppressant of the amphetamine family. Developed in 1962, it...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

dimethylserotonin or as 5-hydroxy-N,N-dimethyltryptamine (5-HO-DMT), is a serotonergic psychedelic of the tryptamine family. It is a derivative of the psychedelic...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

in the mammalian brain, and regulates the activity of dopaminergic, serotonergic and glutamatergic systems. In the human gut, bacteria convert dietary...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

neurotransmitter and hormone and the endogenous ligand of the serotonin receptors. Serotonergic psychedelics such as tryptamines (e.g., psilocybin, psilocin, DMTTooltip...

the transporters. List of antidepressants Noradrenergic and specific serotonergic antidepressant Shaw, W. L. (1980-01-01). "The comparative safety of mianserin...

generic name (help) Bero, Lisa (1987). The interaction of opioid and serotonergic systems regulation prolactin secretion in the developing rat (PhD dissertation)...

1-Valeryl-N,N-diethyllysergamide Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen Legal status Legal status AU: S8 (Controlled...

water (+)-sabinene synthase, an enzyme Serotonin syndrome, due to some serotonergic medications Sjögren's syndrome, an autoimmune disease Sweet's syndrome...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

efavirenz, glaucine, IHCH-7113, MK-212, quipazine, RH-34) For a full list of serotonergic psychedelics, see the navbox here and the list here instead. Dissociatives...

effects of serotonergic, noradrenergic or dual reuptake inhibitors in the carrageenan test in rats: evidence for synergism between serotonergic and noradrenergic...

methylisopropylamide (1-propanoyl-MiPLA), is a designer drug and presumed serotonergic psychedelic of the lysergamide family related to lysergic acid diethylamide...

5-dimethoxyphenethylamine Drug class Serotonin 5-HT2A receptor partial agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name 2-(4-ethoxy-3...

5-HT2A receptor signalling efficacy and not biased agonism differentiates serotonergic psychedelic from non-psychedelic drugs". Br J Pharmacol bph.70109. doi:10...

screening the receptor and other target interactions of 35 different serotonergic psychedelics and related psychoactive drugs in 2010. He selected these...

serotonin 5-HT2A receptor. Similarly to psilocybin, psilocin, and other serotonergic psychedelics, 4-AcO-DMT produces the head-twitch response, a behavioral...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

basis for sleep bruxism and sleep apnea, as well as the role of the serotonergic and dopaminergic pathways in the etiology of sleep bruxism and sleep...

based on their pharmacological mechanisms as psychedelics (which are serotonergic), dissociatives (which are generally antiglutamatergic), or deliriants...

generally avoided because of monoamine-releasing activity, including serotonergic activity. Cocaine is also avoided because of potent monoamine reuptake...

norepinephrine releasing agent (SNRA). The drug shows greatly reduced serotonergic neurotoxicity in comparison to MDMA in animals, although it still shows...

highly selective serotonin releasing agent (SSRA) and does not produce serotonergic neurotoxicity in rodents. These data appear to confer a profile of MMA...

concentrations of serotonin and dopamine, and, therefore, an increase in serotonergic and dopaminergic neurotransmission. A closely related type of drug is...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

proliferation and insulin secretion; PRL, prolactin; PRL secretion is induced by serotonergic hypothalamic signaling; Trp, tryptophan, and Leu, leucine, essential...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

demonstrated therapeutic effects include ketamine, MDMA, scopolamine, and the serotonergic psychedelics, including LSD, psilocin (the active metabolite of psilocybin)...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Tetrahydropalmatine Shoji N, Umeyama A, Takemoto T, Ohizumi Y (April 1984). "Serotonergic receptor antagonist from Nandina domestica Thunberg". Journal of Pharmaceutical...

against methylenedioxymethamphetamine (MDMA)-induced serotonergic neurotoxicity in rodents. The serotonergic neurotoxicity of MDMA appears to be dependent on...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

during long-term use. The norpethidine metabolite was found to have serotonergic effects, so pethidine could, unlike most opioids, increase the risk of...

Quipazine, also known as 1-(2-quinolinyl)piperazine (2-QP), is a serotonergic drug of the arylpiperazine family and an analogue of 1-(2-pyridinyl)piperazine...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

EA1319; 3C-Mescaline; 3C-M Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen; Serotonin 5-HT2A receptor agonist ATC code...

is not expected to cause serotonin toxicity by itself unless another serotonergic drug with clinically significant serotonin reuptake inhibition or serotonin-releasing...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

these substances in synaptic clefts and helping enhance satiety; the serotonergic action, in particular, is thought to influence appetite. Older anorectic...

pepper (and of other plants in the family Piperaceae). Ilepcimide has serotonergic activity. Black pepper Ganellin CR, Triggle DJ (21 November 1996). Dictionary...

SL88.0338 is a serotonergic drug with a benzoylpiperidine structure, which is used in scientific research. It acts as a potent and selective 5-HT1A receptor...

names 2C-C-NBOH; NBOH-2CC Routes of administration Sublingual Drug class Serotonergic psychedelic; Hallucinogen Legal status Legal status BR: Class F2 (Prohibited...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

(5-MeO-iPALT), is a serotonin receptor agonist and serotonergic psychedelic of the tryptamine and 5-methoxytryptamine families which...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status AU:...

thought to be specifically responsible for the hallucinogenic effects of serotonergic psychedelics.[citation needed] 4-HO-DiPT produces the head-twitch response...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

behavior. For example, abnormal hormonal responses to challenges with serotonergic agents have been observed during acute illness, but not recovery. Nevertheless...

blunting than SSRIs and SNRIs. Vortioxetine used in combination with other serotonergic drugs such as MAOIs or SSRIs may result in serotonin syndrome. Vortioxetine...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

GSK-958108 is a serotonergic drug derived from the phenylpiperazine family which acts as a potent and selective 5-HT1A receptor antagonist, and has been...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

antagonist and reuptake inhibitor – Class of drug Noradrenergic and specific serotonergic antidepressant – Class of antidepressants Olver JS, Burrows GD, Norman...

IHCH-7113 is a serotonin 5-HT2A receptor agonist and serotonergic psychedelic of the pyridopyrroloquinoxaline family. It was derived by structural simplification...

MYCO-005 Clinical data Other names MYCO005 Drug class Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen...

Routes of administration Oral Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name (6aR,9R)-N...

Receptor/signaling modulators • Adrenergics • Dopaminergics • Melatonergics • Serotonergics • Monoamine reuptake inhibitors • Monoamine releasing agents • Monoamine...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

needed] Mechanistically, α2 blockers increase adrenergic, dopaminergic and serotonergic neurotransmitters and induce insulin secretion, decreasing blood sugar...

N,N-dihexyltryptamine, is a drug of the tryptamine family related to serotonergic psychedelics like dimethyltryptamine (DMT). It is an analogue in the...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Moclobemide nevertheless has clinically important interactions with some serotonergic and sympathomimetic drugs. Moclobemide was first introduced for medical...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

among many others. The active compounds in these snuffs include the serotonergic psychedelics bufotenin (5-HO-DMT), dimethyltryptamine (DMT), and 5-MeO-DMT...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

majorly altered states of consciousness. Psychedelics, also known as serotonergic psychedelics or classical hallucinogens, are serotonin 5-HT2A receptor...

class Serotonin receptor modulator; Serotonin 5-HT2 receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Lightman, Sl; Nutt, Dj (June 2009). "That warm fuzzy feeling: brain serotonergic neurons and the regulation of emotion". Journal of Psychopharmacology...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

killers" or hallucinogen antidotes in aborting or shortening the effects of serotonergic psychedelics like psilocybin, LSD, and mescaline. Ketanserin, risperidone...

neurons. This results in the conversion of levodopa into dopamine in serotonergic neurons (which cannot re-uptake dopamine and have no proper regulatory...

1-(4-(Trimethylsilyl)benzoyl)-LSD Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Chemical and physical data Formula...

Receptor/signaling modulators • Adrenergics • Dopaminergics • Melatonergics • Serotonergics • Monoamine reuptake inhibitors • Monoamine releasing agents • Monoamine...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

efavirenz, glaucine, IHCH-7113, MK-212, quipazine, RH-34) For a full list of serotonergic psychedelics, see the navbox here and the list here instead. Dissociatives...

Serotonin 5-HT2 receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen; Stimulant; Cognitive enhancer Legal status...

5-dimethoxyphenethylamine, is a serotonin receptor agonist and putative serotonergic psychedelic of the phenethylamine and 2C families. The active dose of...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

role in the regulation of circadian rhythm as research has shown that serotonergic agonism in the SCN results in "phase shifts" in portions of the light-dark...

alternative to MDMA. However, 5-MAPB has been found to be a dose-dependent serotonergic neurotoxin in rodents similarly to MDMA, and might also be a dopaminergic...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

of synaptic vesicle membrane dopaminergic synapse cholinergic synapse serotonergic synapse Biological process ion transport transmembrane transport sodium...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

"Intra-uterine diazepam exposure decreases the number of catecholaminergic and serotonergic neurons of neonate rats". Neuroscience Letters. 795 137014. doi:10.1016/j...

Isopropylidenedioxyamphetamine Drug class Monoamine releasing agent; Entactogen; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name 1-(2,2-dimethyl-1...

family. It is the 1-isopropylated and 6-fluorinated derivative of the serotonergic psychedelic psilocin. The drug is said to be a serotonin 5-HT2A receptor...

of administration Oral Drug class Serotonin 5-HT2 receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

N-diethyllysergamide; SYN-L-229 Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

agent of serotonin, norepinephrine, and dopamine. It produces much less serotonergic neurotoxicity than MDMA in animals. 5-IAI was developed in the 1990s...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Routes of administration Smoking Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Onset of...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

strong serotonin receptor blocking effects make it useful for treating serotonergic crisis such as serotonin syndrome. Dextromethorphan for its part is widely...

potential for serious drug interactions. These include concomitant use with serotonergic agents like selective serotonin reuptake inhibitors (SSRIs), MDMA, and...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

scale. The extensive serotonergic neurotoxicity of 4-chloroamphetamine (and its brominated derivative), and the increased serotonergic toxicity of 4-methylamphetamine...

of serotonin 5-HT2A receptors in studies. (R)-DOI and several other serotonergic psychedelics, including TCB-2, LSD, and LA-SS-Az, have been found to...

MM-77 is a piperazine derivative which is a serotonergic drug, acting as a potent and selective 5-HT1A receptor antagonist. It is used for research into...

class Serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status AU:...

afterglow phenomenon: a systematic review of subacute effects of classic serotonergic psychedelics". Therapeutic Advances in Psychopharmacology. 13 20451253231172254...

Routes of administration Oral Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name (6aR,9R)-N-ethyl-4...

6,7-Dihydroxytryptamine (6,7-DHT) is a serotonergic neurotoxin of the tryptamine family. It is structurally related to the monoamine neurotransmitter serotonin...

Nassa may refer to: Noradrenergic and specific serotonergic antidepressant or NaSSA Nassa (gastropod) NASSA, Negro American Space Society of Astronauts...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

1186/1746-160X-5-21. PMC 2780385. PMID 19895705. Lambru G, Matharu M (April 2011). "Serotonergic agents in the management of cluster headache". Current Pain and Headache...

2023. Glennon RA, Teitler M, Sanders-Bush E (1992). "Hallucinogens and serotonergic mechanisms" (PDF). NIDA Res Monogr. 119: 131–135. PMID 1435968. Archived...

N-Acetylcysteine (NAC) Naltrexone (low-dose) Probiotics and prebiotics Serotonergic psychedelics (e.g., psilocybin) Sleep aids (e.g., orexin receptor antagonists...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

for the treatment of prostate cancer. Due to its action on both the serotonergic and adrenergic systems, venlafaxine is also used as a treatment to reduce...

1-[4-(Trifluoromethyl)phenyl]piperazine (pTFMPP) is a serotonergic releasing agent. It is rarely encountered as a designer drug but is much less common...

study. Recent evidence suggests that changes in both dopaminergic and serotonergic tone alter running-wheel activity. For example, one study in mice has...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Receptor/signaling modulators • Adrenergics • Dopaminergics • Melatonergics • Serotonergics • Monoamine reuptake inhibitors • Monoamine releasing agents • Monoamine...

class Serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

and putative serotonergic psychedelic. It is the O-pivalyl analogue of the naturally occurring but peripherally selective serotonergic tryptamine bufotenine...

synthetic prodrug of the non-selective serotonin receptor agonist and serotonergic psychedelic psilocin which is under development for the treatment of...

provoked or becomes frustrated. Several animal studies note the role of serotonergic functioning in impulsive aggression and antisocial behavior. However...

Receptor/signaling modulators • Monoamine releasing agents • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Many years after being withdrawn, αET was also determined to produce serotonergic neurotoxicity, similarly to MDMA and various other SNDRAs; the same is...

Nonproprietary Name), also known as 2-bromolisuride, is an antidopaminergic and serotonergic agent of the ergoline group which was described as having atypical antipsychotic...

isotryptamine-LSD, is a serotonin receptor modulator, psychoplastogen, and serotonergic psychedelic related to lysergic acid diethylamide (LSD). It is the analogue...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

(ARAS), which includes noradrenergic, dopaminergic, histaminergic, and serotonergic nuclei that promote wakefulness. Amphetamine's therapeutic mode of action...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

4-methylenedioxyamphetamine; DMMDA; DMMDA-1 Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status CA:...

agonists) (e.g., progesterone, medroxyprogesterone acetate) Propofol Serotonergic psychedelics (e.g., psilocybin, lysergic acid diethylamide (LSD), dimethyltryptamine...

extracellular concentrations of serotonin and, therefore, an increase in serotonergic neurotransmission. It is a type of monoamine reuptake inhibitor (MRI);...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

5-DMPEA or 4-BnO-3,5-DMPEA), is a serotonin receptor agonist and possible serotonergic psychedelic of the phenethylamine and scaline families. According to...

NORLAD; NOR-LAD; 6-Nor-LSD Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name (6aR,9R)-N...

administration Oral, others Drug class Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status DE:...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

N-Benzyl-2C-B; NB-2C-B Drug class Serotonin 5-HT2 receptor agonist; Serotonergic psychedelic; Hallucinogen Legal status Legal status In general Unscheduled...

will chemically stimulate neurons. In fact, kainate seems to regulate serotonergic activity in the vertebrate retina. Electrical stimulation of designated...

efavirenz, glaucine, IHCH-7113, MK-212, quipazine, RH-34) For a full list of serotonergic psychedelics, see the navbox here and the list here instead. Dissociatives...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

O-Propionyl-4-HO-MET; O-Propionylmetocin Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

families that was never marketed. It is closely structurally related to serotonergic psychedelics and entactogens like α-methyltryptamine (αMT) and α-ethyltryptamine...

Serotonin 5-HT2 receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status BR:...

irreversible sexual dysfunction at approximately 0.46% of patients treated with serotonergic antidepressants, including SSRIs, though the actual prevalence remains...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

2-aminoindane analogue of fenfluramine and has approximately 50% of the serotonergic neurotoxicity in comparison. Substituted 2-aminoindane 5-Trifluoromethyl-2-aminoindane...

isotryptamine homologue of α-methyltryptamine (αMT), which is a more well-known serotonergic psychedelic, entactogen, and stimulant of the tryptamine family with...

irreversible sexual dysfunction at approximately 0.46% of patients treated with serotonergic antidepressants, including SNRIs, though the actual prevalence remains...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

1-(Cyclopropylmethanoyl)-LSD; 1cP; Curie Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen Legal status Legal status AU: S9 (Prohibited...

DOPEGAL DSP-4 MDA (tenamfetamine) Oxidopamine (6-OHDA) Xylamine V-61 Serotonergic 2′-NH2-MPTP (2′-amino-MPTP) 2,4-DCA 2,4,5-THA 2,4,5-THMA pCPE 3-CA 3...

psilocin; Decadeuteropsilocin Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen Pharmacokinetic data Onset of action <15 minutes...

addition to the preceding, the serotonin 5-HT2 receptor agonist and serotonergic psychedelic 25H-NBOMe has been found to attenuate sepsis-associated depressive-like...

Serotonin 5-HT2 receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen Legal status Legal status DE: NpSG (Industrial...

lesser extent, of the 5-HT2A (pKi = 6.0) receptor. In addition to its serotonergic properties, oxaflozane may also produce anticholinergic side effects...

(2-MeOPP), is a phenylpiperazine derivative which is known to act as a serotonergic agent. Along with various other phenylpiperazines, like benzylpiperazine...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name (6aR,9R)-N...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

tetracyclic antidepressant (TeCA) that acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). It was launched in 1989 for the treatment of...

DOPEGAL DSP-4 MDA (tenamfetamine) Oxidopamine (6-OHDA) Xylamine V-61 Serotonergic 2′-NH2-MPTP (2′-amino-MPTP) 2,4-DCA 2,4,5-THA 2,4,5-THMA pCPE 3-CA 3...

theory – Theory of cognitive development in early humans Trip killer § Serotonergic psychedelic antidotes Also known as psilocybin-containing mushrooms,...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

depressants (such as benzodiazepines, opioids, and alcohol) and agents with serotonergic activity. Additionally, individuals with genetic variations leading to...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

tropomyosin receptor kinase B (TrkB) in the hippocampus, and rapidly activates serotonergic and dopaminergic brain systems. Accordingly, it has been found to produce...

Efavirenz produces the head-twitch response, a behavioral proxy of serotonergic psychedelic effects, in animals, and can partially substitute for LSD...

possible exception of agomelatine, which acts on a dual melatonergic-serotonergic pathway. Despite the success of the monoamine hypothesis it has a number...

also be an adverse drug reaction, such as after ingestion of potent serotonergic drugs, where clonus strongly predicts imminent serotonin toxicity (serotonin...

produces psychedelic effects, it is not used as frequently as other serotonergic psychedelics due to its effects on the gastrointestinal tract via 5-HT3...

isotryptamine homologue of dimethyltryptamine (DMT), a more well-known serotonergic psychedelic of the tryptamine family, and represents a small structural...

(2024-04-15). "Metronidazole-induced neurotoxicity: Possible central serotonergic and noradrenergic system involvement". Medical and Pharmaceutical Journal...

Receptor/signaling modulators • Monoamine releasing agents • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

Non-selective serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

simplified lysergamide which is closely related to the highly potent serotonergic psychedelic lysergic acid diethylamide (LSD). It is specifically the...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Routes of administration Oral Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name (6aR...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Non-selective serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status DE:...

N-diisopropyllysergamide or as lysergic acid diisopropylamide, is a putative serotonergic psychedelic of the lysergamide family related to lysergic acid diethylamide...

names 4-HO-αMT; 4-HO-AMT; MP-14 Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status Uncontrolled...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

company that is developing serotonin 5-HT2A receptor agonists related to serotonergic psychedelics as novel anti-inflammatory drugs to treat inflammatory diseases...

XC-130 Yohimbine See also: Receptor/signaling modulators Adrenergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

DOPEGAL DSP-4 MDA (tenamfetamine) Oxidopamine (6-OHDA) Xylamine V-61 Serotonergic 2′-NH2-MPTP (2′-amino-MPTP) 2,4-DCA 2,4,5-THA 2,4,5-THMA pCPE 3-CA 3...

imagination. An inhibitory system involving the thalamus, likely involving serotonergic neurons, inhibits imaginary perceptions from becoming too activated so...

releasing agent; Serotonin 5-HT2 receptor agonist; Entactogen; Serotonergic psychedelic Identifiers IUPAC name 1-(1-benzothiophen-3-yl)propan-2-amine...

Allain H, Vasar E, Bourin M (February 2001). "Role of dopaminergic and serotonergic systems on behavioral stimulatory effects of low-dose alprazolam and...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

agonist, and as a weak monoamine oxidase inhibitor. It may also produce serotonergic neurotoxicity. αET is a substituted tryptamine and is closely related...

Non-selective serotonin receptor agonist; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name...

disorders. One of its indications is to block the hallucinogenic effects of serotonergic psychedelics, for instance to abort psychedelic experiences early or...

by Alexander Shulgin and others, that the hallucinogenic effects of serotonergic psychedelics like DOM might be due to formation of neurotoxic metabolites...

v t e Antimigraine preparations (N02C) Analgesic/abortive Serotonergics Ergolines Dihydroergocryptine Dihydroergotamine Ergotamine (+caffeine, +chlorcyclizine/caffeine)...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen Legal status Legal status DE: NpSG (Industrial...

symptoms in men withdrawn from placebo treatment. The lack of chronic serotonergic stimulation with on-demand dapoxetine minimizes the potentiation action...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Receptor/signaling modulators • Monoamine releasing agents • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

is not well understood, but it is speculated to selectively destroy serotonergic neurons, in a manner similar to the dopaminergic neurotoxicity of 6-hydroxydopamine...

of, is an action that could in theory cancel out the hypothetical serotonergically-mediated appetite suppressant effects of the compound. However, this...

activity, especially serotonergic opioid analgesics such as meperidine (pethidine) and tramadol. Other opioids listed as serotonergic or uncertain-risk include...

and the serotonin 5-HT1B receptor (Ki = 1,050 nM). The drug produces serotonergic peripheral effects in animals, shows similar metabolism and metabolic...

(PMMA), also known as 4-methoxy-N-methylamphetamine (4-MMA), is a serotonergic drug of the amphetamine family related to para-methoxyamphetamine (PMA)...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

product of haloperidol. The agent is specifically a dopaminergic and serotonergic neurotoxin. HPTP is a prodrug of HPP+, which mediates its monoaminergic...

of administration Oral Drug class Serotonin 5-HT2 receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Legal status Legal status BR:...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

4-Propylamphetamine Clinical data Other names 4-PrA; para-Propylamphetamine Drug class serotonergic agent; psychedelic ATC code None Identifiers IUPAC name...

that emerged many decades later with intense scientific research into serotonergic psychedelics. For example: Baudelaire's cycle of reflections on the drug...

"ecstasy") and its stereoisomers as reinforcers in rhesus monkeys: serotonergic involvement". Psychopharmacology (Berl). 161 (4): 356–364. doi:10...

Receptor/signaling modulators • Monoamine releasing agents • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

CT-4201 is a serotonergic psychedelic which is under development for the treatment of major depressive disorder. It is a prodrug of the tryptamine psychedelic...

Dexfenfluramine, formerly sold under the brand name Redux, is a serotonergic drug that was used as an appetite suppressant to promote weight loss. It is...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers IUPAC name (S)-2-(8...

behavioural functions within the brain. They receive inputs from dopaminergic, serotonergic, noradrenergic, and cholinergic cell groups that modulate information...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

injection, intramuscular injection Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Identifiers PubChem CID 10241628...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

5-Dimethoxy-4-phenylthioamphetamine; 4-PhS-DMA Routes of administration Oral Drug class Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

v t e Antimigraine preparations (N02C) Analgesic/abortive Serotonergics Ergolines Dihydroergocryptine Dihydroergotamine Ergotamine (+caffeine, +chlorcyclizine/caffeine)...

Smith CJ, Stevens AL, Sylvers P (2005). "Psychological, autonomic, and serotonergic correlates of parasuicide among adolescent girls". Development and Psychopathology...

class Serotonin receptor modulator; Serotonin 5-HT2A receptor agonist; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Amineptine‡ Bupropion Nomifensine‡ NaSSAsTooltip Noradrenergic and specific serotonergic antidepressants Mianserin Mirtazapine Setiptiline SARIsTooltip Serotonin...

dextrorotary and levorotary enantiomers displayed receptor affinity for the serotonergic 5-HT1A and 5-HT2B subtypes, though direct binding to the serotonin transporter...

aggression. These aggressive reactions may be caused by a disinhibiting serotonergic mechanism. Paradoxical effects of benzodiazepines appear to be dose-related...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

inhibitor Renin inhibitor Selective glucocorticoid receptor modulator Serotonergic Statin – HMG-CoA reductase inhibitor This type of categorisation of drugs...

Combining dextromethorphan with other serotonergic drugs could possibly cause serotonin syndrome, an excess of serotonergic activity in the CNS and peripheral...

Experimental serotonergic drug...

Routes of administration Oral Drug class Serotonin receptor modulator; Serotonergic psychedelic; Hallucinogen ATC code None Pharmacokinetic data Duration...

Aspirin Barbiturates Benzodiazepines Cocaine Lithium Opioids Paracetamol Serotonergic substances Tricyclic antidepressants Cardiovascular Digoxin Dipyridamole...

such as antidepressants, that increase serotonergic tone in brain stem structures. Overall, the serotonergic system is least active during sleep and...

Diarylmethanes Ethylenediamines Tricyclics Dibenzocycloheptenes Hallucinogens Serotonergic psychedelics/serotonin 5-HT2A receptor agonists: Arylpiperazines Phenylpiperazines...

Xibenolol Xipranolol See also: Receptor/signaling modulators Dopaminergics Serotonergics Monoamine reuptake inhibitors Monoamine releasing agents Monoamine metabolism...

Receptor/signaling modulators • Monoamine reuptake inhibitors • Adrenergics • Dopaminergics • Serotonergics • Monoamine metabolism modulators • Monoamine neurotoxins...

meta-analysis showed that benzodiazepines are significantly more effective than serotonergic agents, regardless of treatment length. More research is needed, but...

(ergometrine), and ergotamine, among others. Although not technically a serotonergic psychedelic, the oneirogen ibogaine, a constituent of Tabernanthe iboga...

Histamine receptor agonist Histamine receptor antagonist (H1 H2 H3) Serotonergic Serotonin receptor agonist Serotonin receptor antagonist (5-HT3) Serotonin...

DOPEGAL DSP-4 MDA (tenamfetamine) Oxidopamine (6-OHDA) Xylamine V-61 Serotonergic 2′-NH2-MPTP (2′-amino-MPTP) 2,4-DCA 2,4,5-THA 2,4,5-THMA pCPE 3-CA 3...