Enfubirtida

Enfubirtida
Formula kimikoaC204H301N51O64
Motakonposatu kimiko
Masa molekularra4.491,193 Da
Erabilera
Konposatu aktiboaFuzeon (en) Itzuli
Tratatzen duHartutako Immuno Eskasiaren Sindromea eta HIV infection (en) Itzuli
HaurdunaldiaAustralian pregnancy category B2 (en) Itzuli eta US pregnancy category B (en) Itzuli
RolaHIV fusion inhibitors (en) Itzuli eta Bakterizida
Identifikatzaileak
InChlKeyPEASPLKKXBYDKL-FXEVSJAOSA-N
CAS zenbakia159519-65-0
ChemSpider16743716
PubChem16130199, 126456160 eta 16157631
Reaxys9612670, 8758835, 11360774, 9384544 eta 11023586
Gmelin608828
ChEMBLCHEMBL525076
EC zenbakia641-385-0
ECHA100.169.201
MeSHD000077560
RxNorm139896
UNII19OWO1T3ZE
NDF-RTN0000148793
KEGGD02499
Ohar medikoa
Ohar medikoa
Oharra: Wikipediak ez du mediku aholkurik ematen. Tratamendua behar duzula uste baduzu, jo ezazu sendagilearengana.

Enfubirtida[1] fusioaren inhibitzaileen familiako antirretrobirala da. Trimeris enpresak sortua, GIB-1 birusarekin infektatutako pazienteetan erabili dute, tratamendu antirretrobiral oso gogorra jaso dutenean eta birusak beste medikamentu batzuekiko erresistentzia garatu duenean.[2]

Erreferentziak

  1. Euskalterm: [Farmakoak Hiztegia] [2022]
  2. Lalezari, JP; Eron, JJ; Carlson, M; Cohen, C; Dejesus, E; Arduino, RC; Gallant, JE; Volberding, P et al.. (2003). «A phase II clinical study of the long-term safety and antiviral activity of enfuvirtide-based antiretroviral therapy» AIDS (Londres) 17 (5): 691–8.  doi:10.1097/01.aids.0000050825.06065.84. PMID 12646792..

Kanpo estekak


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