Search Results: KV1.3

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KCNA3
Kamis, 2025-09-25 05:35:28

Potassium voltage-gated channel, shaker-related subfamily, member 3, also known as KCNA3 or Kv1.3, is a protein that in humans is encoded by the KCNA3 gene....

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Clofazimine
Jumat, 2026-05-22 09:26:47

diabetes. Because the Kv1.3-high effector memory T cells (TEM) are actively involved in the development of these diseases, and Kv1.3 activity is essential...

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Kv1.1
Jumat, 2026-04-24 00:53:31

Potassium voltage-gated channel subfamily A member 1 also known as Kv1.1 is a shaker related voltage-gated potassium channel that in humans is encoded...

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Stichodactyla toxin
Rabu, 2026-08-12 00:35:48

mouse Kv1.3 external vestibule (corresponds to Asp433 in human Kv1.3). Several ShK analogues have been generated to enhance specificity for the Kv1.3 channel...

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Pi5
Rabu, 2025-06-11 06:27:33

the African emperor scorpion Pandinus imperator. Pi5 inhibits human Kv1.2 and Kv1.3 channels as well as Drosophila Shaker B potassium channels. Pi5 is...

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Pandinus imperator (Pi3) toxin
Selasa, 2025-06-24 09:53:41

potassium channel, Kv1.3 and is closely related to another peptide found in the venom, Pi2. Pi3 toxin stands for Pandinus imperator-3 toxin. It is also...

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Hg1 (toxin)
Rabu, 2026-03-18 11:41:17

it selectively inhibits the potassium channel Kv1.3 and, with a lower affinity, channels Kv1.1 and Kv1.2. The Hg1 toxin is named after the Mexican scorpion...

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Human uses of scorpions
Kamis, 2025-11-06 00:47:13

peptides. An important physiological role of the KCNA3 channel, also known as KV1.3, is to help maintain large electrical gradients for the sustained transport...

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Ts15
Senin, 2021-10-25 03:01:35

It targets voltage-gated potassium channels, primarily the subtypes Kv1.2 and Kv1.3. Ts15 can be isolated from the venom of Tityus serrulatus, otherwise...

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BmP02
Sabtu, 2026-06-13 05:24:21

martensi Karsch (BmK) scorpion. The toxin acts on potassium channels, blocking Kv1.3 and slowing the deactivation of Kv4.2. BmP02 is not toxic to humans or mice...

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BF9
Sabtu, 2025-05-24 01:45:19

inhibit both serine proteases and potassium channels (more specifically the Kv1.3 channel). Venom basic protease inhibitor IX, also named BF9, is derived...

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Ctri9577
Senin, 2026-06-22 19:18:15

a potent blocker of the voltage-gated potassium channel Kv1.3, and a gating modifier of Kv4.3 channels. The Ctri9577 toxin is a component of the venom...

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LmKTT-1a
Minggu, 2025-09-28 07:24:22

toxin, it both inhibits trypsin activity and blocks Kv1 channels with a weak selectivity towards Kv1.3 channels. The LmKTT-1a toxin was first identified...

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Kaliotoxin
Rabu, 2026-07-29 09:26:22

Kaliotoxin (KTX) inhibits potassium flux through the Kv1.3 voltage-gated potassium channel and calcium-activated potassium channels by physically blocking...

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LmKTx10
Selasa, 2026-01-27 05:33:17

channels of the family Kv1. It has a higher selectivity for the Kv1.3 potassium channel (KCNA3), compared to other channels in the Kv1 family. The Name LmKTx10...

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Hefutoxin
Jumat, 2026-04-10 22:21:45

unique structure. It blocks the potassium channels Kv1.2 and Kv1.3 and slows the activation of Kv1.3. The kappa- Hefutoxin 1 and 2 (κ- hefutoxin1/2) are...

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Gary Desir
Kamis, 2025-10-16 00:54:30

Li, Yanling Wu, and Gary V. Desir. The voltage-gated potassium channel Kv1.3 regulates peripheral insulin sensitivity Jianchao Xu, Peili Wang, Yanyan...

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Spinoxin
Minggu, 2026-02-01 09:07:38

effects by inhibiting voltage-gated potassium channels, specifically Kv1.2 and Kv1.3. Spinoxin is isolated from the venom of the Malaysian black scorpion...

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Margatoxin
Sabtu, 2025-06-14 04:28:55

Margatoxin (MgTX) is a peptide that selectively inhibits Kv1.3 voltage-dependent potassium channels. It is found in the venom of Centruroides margaritatus...

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Cm28
Kamis, 2025-10-16 01:38:59

margaritatus, selectively blocks voltage-gated potassium channels KV1.2 and KV1.3 with high affinity. It also suppresses the activation of human CD4+...

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Psora-4
Senin, 2026-06-08 16:39:08

Psora-4 is an experimental drug that acts as a selective inhibitor of the Kv1.3 potassium channel. It has immunomodulatory effects, suppressing the proliferation...

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ImKTX58
Minggu, 2025-11-16 18:17:52

the lesser brown scorpion). It is known for its selective inhibition of Kv1.3 channels, on which it acts as a pore-blocker. The name of ImKTX58 stems...

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Hongotoxin
Kamis, 2025-07-17 00:33:35

Shaker-type (Kv1) K+ channels. HgTX1 shows high affinity with Kv1.1, Kv1.2, Kv1.3 voltage-gated potassium channels, but much lower affinity with Kv1.6 (see...

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OdK2
Sabtu, 2026-05-16 01:51:56

α-KTx family, and selectively blocks the voltage-gated potassium channel Kv1.3 (KCNA3). OdK2 is an acronym for the species of origin, the substrate of...

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MeuKTX
Minggu, 2021-10-24 04:13:53

eupeus. This short-chain peptide blocks potassium channels, such as Kv1.1, Kv1.2 and Kv1.3. MeuKTX is a neurotoxin found in the venom of the scorpion Mesobuthus...

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BscTx3
Senin, 2024-12-23 07:08:30

potassium channels Kv1.1, Kv1.2, Kv1.3, Kv1.6 as well as Drosophila Shaker IR channels. The IC50 values for these channels are 172.59 nM for Kv1.2/KCNA2, 2245...

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Cvill7
Sabtu, 2025-12-20 15:47:02

toxins. Particularly, Cvill7 exerts a high affinity for Kv1.2, with weaker effects on Kv1.1 and Kv1.3. | colspan="2" |Cvill7 |- |Superfamily |Scorpion toxins...

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Hemitoxin
Kamis, 2023-11-02 21:24:25

Iranian scorpion Hemiscorpius lepturus, which reversibly blocks Kv1.1, Kv1.2 and Kv1.3 voltage-gated K+ channels. HTX is a neurotoxin derived from the...

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HsTx1
Minggu, 2025-08-31 14:13:54

the rat Kv1.3 voltage-gated potassium channel. HsTx1 stands for Heterometrus spinifer Toxin 1. The systematic name for this toxin is α-KTx 6.3. HsTx1 is...

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Tst26
Selasa, 2025-05-27 12:45:03

stigmurus, a species of Brazilian scorpion. Tst26 selectively blocks Kv1.2 and Kv1.3 channels. Tst26 is named after the species it was discovered from and...

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BmK NSPK
Kamis, 2024-06-06 07:45:16

with BmKTX (Buthus martensii kaliotoxin), which is a previously discovered Kv1.3 channel blocker, BmK NSPK showed 79% sequence homology. Furthermore, BmKTX...

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OSK3
Sabtu, 2025-10-11 01:35:39

subfamily and targets the voltage-gated potassium channels KCNA2 (Kv1.2), and KCNA3 (Kv1.3). OSK3 is secreted from the venom gland of Orthochirus scrobiculosus...

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Pandinus imperator toxin
Kamis, 2025-09-18 03:18:17

voltage-gated potassium channel Kv1.2. at low concentrations (IC50 8.0 ± 5 pM). No significant effects have been observed on Kv1.1 and Kv1.3 channels at concentrations...

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Anuroctoxin
Senin, 2024-12-23 07:08:38

of potassium channel acting peptides. It is a high-affinity blocker of Kv1.3 channels. Anuroctoxin is a peptide which is derived from the scorpion Anuroctonus...

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BmKTX
Senin, 2025-11-03 11:14:00

BmKTX (alpha-KTx 3.6) is a scorpion neurotoxin which blocks the voltage gated potassium channel Kv1.3. The name BmK part of the toxin is derived from the...

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Psoralen
Jumat, 2026-07-24 08:15:56

Heike Wulff (November 2005). "Design of PAP-1, a selective small molecule Kv1.3 blocker, for the suppression of effector memory T cells in autoimmune diseases"...

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Lesional demyelinations of the central nervous system
Kamis, 2026-08-13 08:00:57

Wulff H, Calabresi PA, Allie R, et al. (June 2003). "The voltage-gated Kv1.3 K(+) channel in effector memory T cells as new target for MS". J. Clin....

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BgK
Senin, 2025-11-17 22:15:10

BgK blocks the Kv1.1, Kv1.2, and Kv1.3 channels with similar affinities. IC50 is 6 nM for Kv1.1, 15 nM for Kv1.2, and 10 nM for Kv1.3. Meanwhile, tests...

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Parabutoxin
Sabtu, 2025-06-21 06:28:29

Shaker-related voltage-gated potassium channels members 1,2 and 3 (Kv1.1, Kv1.2 and Kv1.3 channels). These channels have different functions that include...

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Zoltán Takács (toxinologist)
Rabu, 2025-10-01 20:38:22

Suarez-Kurtz G, Koide S, Goldstein SA (2009). "A designer ligand specific for Kv1.3 channels from a scorpion neurotoxin-based library". Proceedings of the National...

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Olivierus martensii
Selasa, 2026-04-21 05:51:36

used in anticancer treatments. BmP02 acts on potassium channels, blocking Kv1.3 and slowing the deactivation of Kv4.2. BmP02 is not toxic to humans or mice...

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Tyrosin-protein kinase Lck
Kamis, 2026-04-16 03:22:52

large tumor suppressor binds to p56lck tyrosine kinase and Shaker type Kv1.3 potassium channel in T lymphocytes". The Journal of Biological Chemistry...

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Developmental bioelectricity
Kamis, 2026-08-13 03:33:23

PMID 26216856. Duque, A.; Gazula, V. R.; Kaczmarek, L. K. (2013). "Expression of Kv1.3 potassium channels regulates density of cortical interneurons". Developmental...

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KCNA5
Rabu, 2025-07-23 22:29:50

voltage-gated channel, shaker-related subfamily, member 5, also known as KCNA5 or Kv1.5, is a protein that in humans is encoded by the KCNA5 gene. Potassium channels...

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KCNA4
Selasa, 2025-07-15 11:20:40

Potassium voltage-gated channel subfamily A member 4 also known as Kv1.4 is a protein that in humans is encoded by the KCNA4 gene. It contributes to the...

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Multiple sclerosis drug pipeline
Selasa, 2026-03-31 11:28:41

suppress myelin-reactive effector memory T cells by blocking voltage-gated Kv1.3 channels in these cells. hydralazine: Due to its ability to damage myelin...

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ImKTx88
Sabtu, 2026-03-28 21:50:53

ImKTx88 is a selective inhibitor of the Kv1 ion channel family that can be isolated from the venom of the Isometrus maculatus (lesser brown scorpion)...

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Markus Sperandio
Senin, 2026-05-25 00:33:43

Deutsche Forschungsgemeinschaft. Retrieved 2026-05-05. "C2: The role of KV1.3 on Ca2+ signalling and neutrophil effector functions". Website of the Transregio...

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Mesobuthus eupeus
Selasa, 2026-05-19 01:05:49

M. martensii, potently inhibits rKv1.1, rKv1.2 and hKv1.3 channels but does not affect rKv1.4, rKv1.5, hKv3.1, rKv4.3, and hERG channels even at high concentrations...

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Maurotoxin
Sabtu, 2026-04-18 16:32:34

channels (IK) Several types of voltage-gated potassium channels (Kv1.1, Kv1.2, Kv1.3 and shaker B) The structural and pharmacological features of MTX...

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Christine Beeton
Kamis, 2026-03-26 02:19:00

the first person able to show the significant benefits of blocking Kv1.1 and Kv1.3 channels with kaliotoxin - a component of scorpion venom - as a preventative...

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List of MeSH codes (D12.776.543)
Jumat, 2025-08-15 03:47:17

311 – kv1.1 potassium channel MeSH D12.776.543.550.425.750.900.124.342 – kv1.2 potassium channel MeSH D12.776.543.550.425.750.900.124.358 – kv1.3 potassium...

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Scaffold protein
Selasa, 2026-03-24 06:08:23

Large Tumor Suppressor Binds to p56 lck Tyrosine Kinase and Shaker Type Kv1.3 Potassium Channel in T Lymphocytes". Journal of Biological Chemistry. 272...

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Voltage-gated potassium channel
Sabtu, 2026-06-20 02:14:05

non-inactivating Kvα1.x - Shaker-related: Kv1.1 (KCNA1), Kv1.2 (KCNA2), Kv1.3 (KCNA3), Kv1.5 (KCNA5), Kv1.6 (KCNA6), Kv1.7 (KCNA7), Kv1.8 (KCNA10) Kvα2.x - Shab-related:...

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Ssm spooky toxin
Minggu, 2026-05-31 09:16:11

(KV7.1, KV7.2, KV7.4, and KV7.5) but it has also been found to inhibit KV1.3 (and the Drosophila homolog shaker), KV2.1 (KCNB1) and KV4 (and its Drosophila...

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Calyx of Held
Minggu, 2026-07-26 08:20:57

present: Kv1.1, Kv1.2, Kv1.3, and Kv7.5. Kv1.1 and Kv1.2 are located in the transition zone between the axon and the terminal, while Kv1.3 Kv7.5 are...

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KCNA2
Senin, 2025-11-17 23:03:52

Potassium voltage-gated channel subfamily A member 2 also known as Kv1.2 is a protein that in humans is encoded by the KCNA2 gene. Potassium channels...

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Jonathan Baell
Rabu, 2026-02-11 01:34:29

"Khellinone Derivatives as Blockers of the Voltage-Gated Potassium Channel Kv1.3: Synthesis and Immunosuppressive Activity". Journal of Medicinal Chemistry...

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DLG1
Sabtu, 2025-12-06 04:34:13

large tumor suppressor binds to p56lck tyrosine kinase and Shaker type Kv1.3 potassium channel in T lymphocytes". The Journal of Biological Chemistry...

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SGK1
Selasa, 2026-02-24 06:07:42

and epithelial K+ channels KCNE1/KCNQ1 Voltage-gated K+ channels Kv1.3, Kv1.5, and Kv4.3 Glutamate Receptors The following carriers and pumps are influenced...

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List of MeSH codes (D12.776.157)
Jumat, 2025-08-15 03:43:00

124 – kv1.1 potassium channel MeSH D12.776.157.530.400.600.900.500.186 – kv1.2 potassium channel MeSH D12.776.157.530.400.600.900.500.217 – kv1.3 potassium...

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KCNA6
Sabtu, 2025-07-19 03:39:09

Potassium voltage-gated channel subfamily A member 6 also known as Kv1.6 is a protein that in humans is encoded by the KCNA6 gene. The protein encoded...

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Stichodactyla helianthus
Selasa, 2026-06-23 12:22:19

Specific Kv1.3 Channel Inhibitor That Suppresses T Cell Mediators of Autoimmune Disease". The Journal of Pharmacology and Experimental Therapeutics. 342 (3):...

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Potassium channel blocker
Selasa, 2026-06-23 13:40:46

voltage-gated Kv2.1 potassium channel currents. a very potent inhibitor of the rat Kv1.3 voltage-gated potassium channel Voigt N, Dobrev D (2016). "Atrial-Selective...

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APEKTx1
Sabtu, 2025-08-30 20:13:03

channel Kv1.1 with no effect on other tested potassium channels (Kv1.2, Kv1.3, Kv1.4, Kv1.5, Kv1.6, Shaker IR, Kv2.1, Kv3.1, Kv4.2 and Kv4.3). APEKTx1...

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Cation channel superfamily
Kamis, 2025-10-02 00:53:46

RYR3 Kvα1.x - Shaker-related: Kv1.1 (KCNA1), Kv1.2 (KCNA2), Kv1.3 (KCNA3), Kv1.5 (KCNA5), Kv1.6 (KCNA6), Kv1.7 (KCNA7), Kv1.8 (KCNA10) Kvα2.x - Shab-related:...

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KCNE2
Selasa, 2025-09-16 05:02:47

forms complexes there with the voltage-gated potassium channel α subunit, Kv1.3. In addition, KCNE2 forms reciprocally regulating tripartite complexes in...

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Gambierol
Minggu, 2025-08-31 14:48:03

especially Kv1.1-1.5 channels and the Kv3.1 channel. Kv1.1-1.5 channels are responsible for repolarization of the membrane potential. The Kv1.3 channel however...

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CboK7
Kamis, 2025-10-16 01:38:43

bonito. It blocks voltage-gated K+ channels, with the highest affinity for Kv1.2 channels. This toxin is known by two names: CboK7 and α-KTx 2.24. The name...

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Episodic ataxia
Selasa, 2025-07-15 11:08:14

encodes the voltage-gated potassium channel KV1.1, are responsible for this subtype of episodic ataxia. KV1.1 is expressed heavily in basket cells and...

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Ts8
Sabtu, 2026-01-31 05:25:58

in three forms, of which Ts8-FragII has a small inhibitory effect on the Kv1.3 channel. The inhibition caused by the neurotoxin Ts8 on Kv4.2 channels increases...

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Heteroscodratoxin-1
Rabu, 2025-05-28 20:36:53

and KV3.4) or delayed rectifier potassium channels (KV1.1, KV1.2, KV1.3, KV1.5, KV1.6, KV1.2/ KV1.5, or KVLQT1), or on sodium and calcium channels has...

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SHC3
Kamis, 2025-12-18 14:33:59

proteins differentially modulate the phosphorylation and biophysics of Kv1.3 ion channel by SRC kinase". The Journal of Biological Chemistry. 277 (15):...

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Ramesses VII
Sabtu, 2026-06-20 14:28:27

was buried in Tomb KV1 upon his death. Finely carved wall reliefs in Ramesses VII's KV1 tomb The Tomb Corridor of Ramesses VII's KV1 tomb His mummy has...

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DUSP3
Kamis, 2025-07-17 00:10:23

Swanson R (Feb 1995). "Confirmation of the assignment of the gene encoding Kv1.3, a voltage-gated potassium channel (KCNA3) to the proximal short arm of...

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KCNAB1
Sabtu, 2025-07-19 13:14:43

large tumor suppressor binds to p56lck tyrosine kinase and Shaker type Kv1.3 potassium channel in T lymphocytes". J. Biol. Chem. 272 (43): 26899–904...

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KCNE4
Senin, 2025-09-29 15:45:50

strongly inhibits Kv1.1 and Kv1.3 channels when co-expressed in HEK cells and in Xenopus laevis oocytes, while leaving Kv1.2 and Kv1.4 currents unaffected...

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Cobatoxin
Sabtu, 2025-09-13 05:11:25

(KTx), which consists of 3 families; α, β, and γ. These 3 families differ in structure. Cobatoxin 1 and 2 both block the Kv1.1 K+-channels in mice and...

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Jackson King V
Sabtu, 2025-06-14 00:45:53

but with dot inlays, no binding, and rosewood fretboard. KV1(Artist Signature Series) The KV1 is a Dave Mustaine signature model and is the first commercially-sold...

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Dave Mustaine
Sabtu, 2026-08-08 21:53:56

meaning it had two of the longer fins from the RR). The reshaped Mustaine KV1 model had slightly shorter fins, Kahler bridge and Seymour Duncan TB-5 bridge...

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Twentieth Dynasty of Egypt
Selasa, 2026-08-04 21:13:55

discovery by Howard Carter in 1922. Ramesses VII's only monument is his tomb, KV1.[citation needed] Almost nothing is known about Ramesses VIII's reign, which...

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Valley of the Kings
Jumat, 2026-08-07 04:26:30

signs for the tombs, providing information and plans of the open tombs. KV1 KV2 KV3 KV4 KV5 KV6 KV7 KV8 KV9 KV10 KV11 KV12 KV13 KV14 KV15 KV16 KV17 KV18...

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List of burials in the Valley of the Kings
Kamis, 2026-07-30 19:13:46

also used to designate tombs located in the West Valley (of the Kings). KV1 KV2 KV3 KV4 KV5 KV6 KV7 KV8 KV9 KV10 KV11 KV12 KV13 KV14 KV15 KV16 KV17 KV18...

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Butantoxin
Kamis, 2025-09-18 20:47:06

blocks the voltage-gated K+ channels Shaker B and Kv1.2, and the Ca2+-activated K+ channels KCa 1.1 and KCa 3.1. Butantoxin is one of multiple toxins isolated...

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Kalicludine
Sabtu, 2025-12-27 20:13:58

Kalicludine (AsKC) is a blocker of the voltage-dependent potassium channel Kv1.2 found in the snakeslocks anemone Anemonia viridis (Anemonia sulcata), which...

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BrMT
Sabtu, 2024-11-23 11:36:04

The disulfide-linked dimer of BrMT possesses inhibitory effects on the Kv1 and Kv4 families of voltage-gated potassium channels. BrMT was first isolated...

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Endocannabinoid system
Sabtu, 2026-06-27 11:21:12

Immunohistochemistry experiments demonstrated that CB1 is co-localized with GIRK and Kv1.4 potassium channels, suggesting that these two may interact in physiological...

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XEN-D0101
Selasa, 2026-06-30 10:15:40

XEN-D0101 is a selective antagonist of the voltage-gated potassium channel Kv1.5. Atrial fibrillation is the main focus of Xention’s drug development, as...

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KCNA10
Sabtu, 2023-03-04 03:33:37

Potassium voltage-gated channel subfamily A member 10 also known as Kv1.8 is a protein that in humans is encoded by the KCNA10 gene. The protein encoded...

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Sisu Nasu
Kamis, 2024-11-14 01:48:53

12 in tail unit. NA-111GT A signal station version. NA-120 GT NA-120 GT KV1 Armoured variant used in UN-operations. NA-122 A version that carries a 120 mm...

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Essential fatty acid
Senin, 2025-12-29 04:01:08

1994). "External blockade of the major cardiac delayed-rectifier K+ channel (Kv1.5) by polyunsaturated fatty acids". Proceedings of the National Academy of...

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Amitriptyline
Selasa, 2026-08-11 22:24:17

(3): 1015–1023. doi:10.1016/S0022-3565(24)35384-4. PMID 10688618. Punke MA, Friederich P (May 2007). "Amitriptyline is a potent blocker of human Kv1.1...

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Kappa-KTx2.5
Senin, 2026-05-11 15:24:44

residue of κ-KTx2.5 interacts with aspartic acid-348 (D348) of Kv1.2 at a distance of 3.7 Å, affecting only one subunit. Lysine-23 (K23) in the toxin likely...

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Kendriya Vidyalaya No. 2, Vizag
Sabtu, 2026-02-21 08:59:53

and one Navy Children School in the Naval Campus. The other three being KV1, NSB; KV Malkapuram; NCS, NSB, Vizag. The school has a fairly big campus...

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Team Secret
Rabu, 2026-07-29 09:52:44

September 19 math was removed from the starting lineup. October 8 Danilo "kv1" Michelini joined. On January 8, 2024, Team Secret announced the formation...

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Sigma-1 receptor
Selasa, 2026-08-11 19:23:23

has been shown to appear in a complex with voltage gated K+ channels (Kv1.4 and Kv1.5), leading to the idea that σ1 receptors are auxiliary subunits. σ1...

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Repolarization
Senin, 2026-04-27 05:53:59

membrane to re-establish the resting potential. The four types are Kv1, Kv2, Kv3 and Kv4. The Kv1 channel primarily influences the repolarization of the axon...

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Activation
Jumat, 2026-01-30 01:25:55

Antonella; Rolland, Jean-Francois; Pessia, Mauro; Imbrici, Paola (2020-04-22). "Kv1.1 Channelopathies: Pathophysiological Mechanisms and Therapeutic Approaches"...

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Morvan's syndrome
Kamis, 2026-08-13 03:34:16

neuromyotonia. It is believed that antibodies to the Shaker-type K+ channels (the Kv1 family) are the type of potassium channel most strongly associated with acquired...

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KCNA7
Minggu, 2022-04-17 10:12:23

Potassium voltage-gated channel subfamily A member 7 also known as Kv1.7 is a protein that in humans is encoded by the KCNA7 gene. The protein encoded...

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Discovery of the tomb of Tutankhamun
Minggu, 2026-07-12 23:31:20

 90–91. Carter & Mace 2003, pp. 91–95. Hoving 1978, p. 87. Frayling 1992, pp. 3–4. Carter & Mace 2003, pp. 95–96. Frayling 1992, pp. 4–5. Reeves 1990, pp...

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Middle Khmer
Minggu, 2026-06-28 01:12:08

pre-Angkor and modern Khmer" (PDF). Pacific Linguistics. 42 (19): 19–38. Retrieved 3 January 2016. Lewitz, Saveros (1967). "La toponymie khmère". Bulletin de l'École...

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Kaamelott: The First Chapter
Rabu, 2026-08-05 06:13:16

"KAAMELOTT - PREMIER VOLET sortira au cinéma le 21 juillet.#KaamelottLeFilm #KV1" (Tweet) – via Twitter. "Kaamelott : Premier Volet sortira en salle le 21...

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GABRA3
Rabu, 2025-10-22 11:33:37

alter chloride permeability of the GABA receptor. At the time of discovery, Kv1.1 mRNA was the only previously known mammalian coding site containing both...

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Palmitoyl acyltransferase
Kamis, 2025-02-13 07:46:34

receptor subunit GluR1 and GluR2, GABAA receptor gamma2 subunit, aquaporin, KV1.1, rhodopsin, beta2-adrenergic receptor, and PSD-95. https://swisspalm.org/enzymes...

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MCD peptide
Jumat, 2024-08-16 16:43:38

characterization of five cloned voltage-gated K+ channels, types Kv1.1, 1.2, 1.3, 1.5, and 3.1, stably expressed in mammalian cell lines". Mol Pharmacol....

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Panchkula
Senin, 2026-08-10 02:46:05

School, Morni Rd Jainendra Public School, Sector 1 Kendriya Vidyalaya No. 1 (KV1), Chandimandir Cantonment Kendriya Vidyalaya No. 2 (KV2), Chandimandir Cantonment...

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4-Aminopyridine
Kamis, 2026-07-23 07:57:08

biophysics.[citation needed] It is a relatively selective blocker of members of Kv1 (Shaker, KCNA) family of voltage-activated K+ channels. However, 4-AP has...

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Rongorongo text K
Senin, 2024-10-28 19:45:14

tablets. There are five lines of glyphs on the recto, a transitional line (Kv1) along the edge, and four lines (Kv2-5) on the verso proper. The first and...

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Heteropodatoxin
Rabu, 2023-07-19 23:33:55

heteropodatoxin-2 blocks the potassium channels Kv4.1, Kv4.2 and Kv4.3, but not Kv1.4, Kv2.1, or Kv3.4. Heterpodatoxin-2 most likely acts as a gating modifier...

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Pandinotoxin
Sabtu, 2025-06-14 04:28:26

channels of the subfamily A member 2 (Kv1.2/KCNA2) [1] and they can reversibly block the shaker B potassium-channels (Kv1.1 sub-family). The residue K27, a...

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Cardiac transient outward potassium current
Sabtu, 2025-11-01 08:44:58

needed] The Ito1 is generated by voltage-gated K+ channels Kv1.4, Kv4.2, and (especially) Kv4.3; these channels undergo ball-and-chain inactivation to terminate...

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Anti-VGKC-complex encephalitis
Minggu, 2026-05-17 22:07:08

detected with the radioimmunoprecipitation assay, only 3 (3%) had antibodies towards the Kv1 subunit of the VGKC channel, 55 (57%) had antibodies against...

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GJC3
Sabtu, 2023-03-04 06:49:56

In both PNS and CNS myelinated axons, Cx29 is precisely colocalized with Kv1.2 voltage-gated K+ channels, where both proteins are concentrated in the...

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Cadherin-2
Selasa, 2026-08-11 17:31:28

that the arrhythmias were likely due to ion channel remodeling and aberrant Kv1.5 channel function. These animals showed a prolonged action potential duration...

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Cortactin
Jumat, 2025-10-31 13:40:40

E, Cachero TG, Morielli AD (October 2002). "Tyrosine phosphorylation of Kv1.2 modulates its interaction with the actin-binding protein cortactin". J...

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Quinidine
Selasa, 2026-06-02 14:49:48

agent. Quinidine also blocks certain voltage-gated potassium channels (e.g., Kv1.4, Kv4.2, hERG, among others), acts as an antimuscarinic and alpha-1 blocker...

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List of unnumbered trans-Neptunian objects
Jumat, 2026-07-03 08:23:58

Spacewatch (691) 76 centaur 35.8 0.62 11 13.6 58.0 albedo: 0.058 MPC · JPL 1996 KV1 21 May 1996 C. A. Trujillo, D. C. Jewitt, J. X. Luu (568) 164 cubewano (hot)...

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KCNAB2
Kamis, 2025-07-17 00:42:22

Coleman SK, Newcombe J, Pryke J, Dolly JO (Aug 1999). "Subunit composition of Kv1 channels in human CNS". J. Neurochem. 73 (2): 849–58. doi:10.1046/j.1471-4159...

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Jackson Y2KV
Sabtu, 2026-06-06 09:35:39

Retrieved 2009-12-21. Jackson Catalog 2001. Tuners are arranged in the classic 3-a side style instead of the usual six a side. These two differences combined...

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List of unnumbered minor planets: 1996
Senin, 2026-07-27 20:52:21

510 m single 66 days 18 Jul 1996 80 Disc.: NEAT/GEODSS MPC · JPL 2 1996 KV1 TNO 7.3 178 km multiple 1996–2016 29 May 2016 27 Disc.: Mauna Kea Obs. LoUTNOs...

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Neuroprotection
Kamis, 2026-08-13 00:13:22

fluid of sporadic amyotrophic lateral sclerosis patients alters Nav1.6 and Kv1.6 channel expression in rat spinal motor neurons". Brain Research. 1255:...

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Saak Ovsepian
Jumat, 2026-06-26 05:07:24

Valerie B O'Leary, Christian Leibold, J Oliver Dolly. "Distinctive role of KV1.1 subunit in the biology and functions of low threshold K+ channels with...

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List of minor planets: 892001–893000
Rabu, 2026-07-01 02:48:00

JN26 — May 14, 2015 Haleakala Pan-STARRS 1  · 2.4 km MPC · JPL 892395 2015 KV1 — April 10, 2015 Haleakala Pan-STARRS 1  · 860 m MPC · JPL 892396 2015 KH10...

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Sulfatide
Kamis, 2026-02-19 23:27:35

number of clusters of sodium channels at the nodes of Ranvier. Additionally, Kv1.2 channels are moved from the paranodal position to the juxtaparanodal position...

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Potassium channel
Sabtu, 2026-06-20 09:34:29

Life Sciences. Vol. 16. Springer. pp. 325–347. doi:10.1007/978-3-319-21756-7_9. ISBN 978-3-319-21755-0. PMID 26860305. indirectly cited from reference number...

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List of cis-regulatory RNA elements
Senin, 2024-10-07 04:32:38

(PIE) UnaL2 LINE 3′ element Vimentin 3′ UTR protein-binding region Voltage-gated potassium-channel Kv1.4 IRES Wingless localisation element 3 (WLE3) xerDC...

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GRIA3
Senin, 2025-10-27 23:16:02

structure is related to that found in K+ channels (e.g., human Kv1.1 channel). The human Kv1.1 channel pre mRNA is also subject to A to I RNA editing. The...

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Pharmacodynamics of spironolactone
Selasa, 2025-12-23 06:16:24

(2005). "Spironolactone and its main metabolite canrenoic acid block hKv1.5, Kv4.3 and Kv7.1+minK channels". British Journal of Pharmacology. 146 (1): 146–161...

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DLG4
Kamis, 2025-07-31 20:47:58

D (November 2002). "N-terminal PDZ-binding domain in Kv1 potassium channels". FEBS Lett. 531 (3): 529–37. Bibcode:2002FEBSL.531..529E. doi:10.1016/S0014-5793(02)03572-X...

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HgeTx1
Senin, 2024-12-23 07:50:44

"Contribution of the functional dyad of animal toxins acting on voltage-gated Kv1-type channels". J Pept Sci. 11 (2): 65–8. doi:10.1002/psc.630. PMID 15635666...

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Tityustoxin
Jumat, 2026-05-22 20:14:34

peptide toxin, interacts with the alpha-dendrotoxin binding site on the cloned Kv1.2 K+ channel". Molecular Pharmacology. 44 (2): 430–436. doi:10.1016/S0026-895X(25)13197-0...

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GRIA2
Senin, 2025-10-27 23:17:06

related to that found in K+ channels, such as the human Kv1.1 channel. The pre-mRNA of the human Kv1.1 channel is also subject to A-to-I RNA editing. Glutamate...

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KCNA2-related disorders
Kamis, 2026-04-09 18:11:06

KCNA2-related disorders are caused by mutations to the Kv1.2 channels encoded by the KCNA2 gene. These neurological disorders are associated with a spectrum...

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LGI1
Jumat, 2026-06-05 08:50:15

Peles E, Buckley C, Lang B, Vincent A (September 2010). "Antibodies to Kv1 potassium channel-complex proteins leucine-rich, glioma inactivated 1 protein...

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Genetically encoded voltage indicator
Selasa, 2026-08-11 23:14:36

fluorescent protein FRET pair, e.g. VSFP1, (2) Single opsin GEVIs, e.g. Arch, (3) Opsin-FP FRET pair GEVIs, e.g. MacQ-mCitrine, (4) single FP with special...

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Index of biophysics articles
Selasa, 2025-09-02 20:37:54

KCNT2 KCNV1 KCNV2 Kenneth Stewart Cole Kim Sung-Hou Kir2.1 Kir2.6 Kir6.2 Kv1.1 KvLQT1 KvLQT2 KvLQT3 L-type calcium channel Lamellar structure Lamellipodium...

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KCNQ1
Jumat, 2026-07-24 04:12:00

Norwegian perspective". Am. J. Med. Genet. 89 (3): 137–146. doi:10.1002/(SICI)1096-8628(19990924)89:3<137::AID-AJMG4>3.0.CO;2-C. PMID 10704188. Gutman GA, Chandy...

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PTPRM
Kamis, 2025-11-20 07:23:37

brain cells. PTPmu has been shown to increase the mRNA of the K+ channel Kv1.5 in cardiac myocytes when CHO cells expressing PTPmu are cultured with cardiac...

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Corticotropin-releasing hormone receptor
Selasa, 2026-08-11 22:51:43

neuronal excitability in the hippocampus by modulating potassium channels (KV1 subfamily), increasing population spike amplitudes through presynaptic mechanisms...

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Gintonin
Jumat, 2025-11-07 11:35:19

(2013). "Activation of lysophosphatidic acid receptor by gintonin inhibits Kv1.2 channel activity: Involvement of tyrosine kinase and receptor protein tyrosine...

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Shaker (gene)
Rabu, 2025-03-26 18:32:21

structure determination of AgTx2-MTX chimera, a new potential blocker for Kv1.2 channel, derived from MTX and AgTx2 scorpion toxins". Protein Science....

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Discrepin
Selasa, 2026-06-09 22:50:11

toxin BmTx3 to its receptor site, where other K+ channel blockers (Kv1-, Kv3.4-, Kv4.2/4.3 family blockers) were unable to compete with this toxin. These...

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List of minor planets: 99001–100000
Senin, 2026-06-15 07:04:15

10, 2002 Palomar NEAT  · 3.2 km MPC · JPL 99787 2002 JM146 — May 15, 2002 Haleakala NEAT V 1.2 km MPC · JPL 99788 2002 KV1 — May 16, 2002 Socorro LINEAR...

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KCNAB3
Rabu, 2024-07-17 05:39:27

Isbrandt D, Pongs O (Feb 1999). "Coexpression of the KCNA3B gene product with Kv1.5 leads to a novel A-type potassium channel". J Biol Chem. 273 (52): 35095–101...

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Antonello Bonci
Selasa, 2026-08-11 15:42:56

TP; Bonci, A (2013). "Dynamic interaction between sigma-1 receptor and Kv1.2 shapes neuronal and behavioral responses to cocaine". Cell. 152 (1–2):...

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Potassium channel tetramerisation domain
Minggu, 2023-12-03 23:24:38

the basis of sequence similarity and function. Four of these subfamilies, Kv1 (Shaker), Kv2 (Shab), Kv3 (Shaw) and Kv4 (Shal), consist of pore-forming...

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AsKC11
Jumat, 2026-05-15 12:34:42

Kir2.1 or the voltage-gated potassium channels, Kv1.1-1.4 channels, and showed a small inhibition of Kv1.6. channels. AsKC11 binding is reversible. For...

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KCND2
Sabtu, 2025-07-19 13:14:47

DF, Fedida D (2002). "N-terminal PDZ-binding domain in Kv1 potassium channels". FEBS Lett. 531 (3): 529–537. doi:10.1016/S0014-5793(02)03572-X. PMID 12435606...

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PTPRA
Kamis, 2025-11-20 06:58:13

participates in the m1 muscarinic acetylcholine receptor-dependent regulation of Kv1.2 channel activity". EMBO J. 18 (1): 109–18. doi:10.1093/emboj/18.1.109....

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Michael G. Hanna
Senin, 2026-05-18 13:50:51

(1999). "A novel mutation in the human voltage-gated potassium channel gene (Kv1.1) associates with episodic ataxia type 1 and sometimes with partial epilepsy"...

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GRIK2
Selasa, 2026-02-24 06:02:47

pore loop structure is similar to that found in K+ channels (e.g. the human Kv1.1 channel, whose pre-mRNA is also subject to A to I RNA editing). The diversity...

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List of minor planets: 732001–733000
Rabu, 2026-04-01 21:22:54

Dictionary of Minor Planet Names. Springer Berlin Heidelberg. ISBN 978-3-540-00238-3. Retrieved 27 July 2016. Schmadel, Lutz D. (2006). Dictionary of Minor...

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Guangxitoxin
Kamis, 2026-04-23 23:29:09

Gaisano HY, Salapatek AM, Backx PH, Wheeler MB (August 2001). "Members of the Kv1 and Kv2 voltage-dependent K(+) channel families regulate insulin secretion"...

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Index of ancient Egypt–related articles
Kamis, 2026-08-13 17:13:23

Kulubnarti church Kulubnarti Kumma (Nubia) Kurna Kurt Sethe Kushite religion KV1 KV2 KV3 KV4 KV5 KV6 KV7 KV8 KV9 KV10 KV11 KV12 KV13 KV14 KV15 KV16 KV18 KV19...

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1st Guards Cavalry Corps
Selasa, 2025-12-23 06:21:25

traditional sabre of the Cossack horsemen. The cavalrymen, along with the T34 and KV1 tanks wielded by the 112th Tank Division battled ferociously against the...

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List of minor planets: 697001–698000
Rabu, 2026-04-01 21:19:33

Dictionary of Minor Planet Names. Springer Berlin Heidelberg. ISBN 978-3-540-00238-3. Retrieved 27 July 2016. Schmadel, Lutz D. (2006). Dictionary of Minor...

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Alpha-actinin-2
Senin, 2026-04-27 12:04:56

Fedida D (July 2003). "SAP97 increases Kv1.5 currents through an indirect N-terminal mechanism". FEBS Letters. 547 (1–3): 205–11. doi:10.1016/S0014-5793(03)00668-9...

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List of minor planets: 426001–427000
Rabu, 2026-04-01 20:51:25

Dictionary of Minor Planet Names. Springer Berlin Heidelberg. ISBN 978-3-540-00238-3. Retrieved 27 July 2016. Schmadel, Lutz D. (2006). Dictionary of Minor...

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Unconventional myosin-Va
Sabtu, 2025-10-04 16:16:29

MYO5B are involved with Kv1.5 (encoded by Potassium voltage-gated channel subfamily A member 5, KCNA5) in the myocytes. Kv1.5 is associated with the...

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List of minor planets: 643001–644000
Rabu, 2026-04-01 21:14:39

Dictionary of Minor Planet Names. Springer Berlin Heidelberg. ISBN 978-3-540-00238-3. Retrieved 27 July 2016. Schmadel, Lutz D. (2006). Dictionary of Minor...

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KCNE1
Selasa, 2025-10-21 19:26:29

co-expressed with the Kv1.1 α subunit in Chinese Hamster ovary (CHO) cells, KCNE1 traps the N-type (rapidly inactivating) Kv1.4 α subunit in the ER/Golgi...

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List of minor planets: 458001–459000
Minggu, 2026-05-10 07:01:47

Dictionary of Minor Planet Names. Springer Berlin Heidelberg. ISBN 978-3-540-00238-3. Retrieved 27 July 2016. Schmadel, Lutz D. (2006). Dictionary of Minor...

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List of minor planets: 508001–509000
Rabu, 2026-04-01 20:59:34

Dictionary of Minor Planet Names. Springer Berlin Heidelberg. ISBN 978-3-540-00238-3. Retrieved 27 July 2016. Schmadel, Lutz D. (2006). Dictionary of Minor...

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AmmTX3
Selasa, 2026-06-02 14:48:10

channels almost completely. A-type potassium currents can be generated by Kv1.4, Kv3.3, Kv3.4, all members of Kv4 and Erg3 channels. The influence of AmmTX3...

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MLC1
Senin, 2026-08-10 09:46:42

homology with the KCNA1 shaker-related voltage-gated potassium channel (Kv1.1). This analysis suggests that MLC1 may be a cation channel.[needs update]...

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Gene therapy for epilepsy
Selasa, 2026-06-23 20:46:52

tone, it is possible to restore balance between inhibition and excitation. Kv1.1 is a voltage-gated potassium channel encoded by the KCNA1 gene. It is widely...

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List of minor planets: 328001–329000
Rabu, 2026-03-25 22:52:59

JPL 328339 2008 KU1 — May 26, 2008 Kitt Peak Spacewatch  · 1.3 km MPC · JPL 328340 2008 KV1 — May 26, 2008 Kitt Peak Spacewatch WIT 1.2 km MPC · JPL 328341...

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KCNE5
Senin, 2025-09-29 21:14:47

KCNQ2/3 or KCNQ5 channel activity, KCNE5 inhibits KCNQ4 in CHO cells but not in oocytes. Although it has no known effects on hERG (Kv11.1) or Kv1.x family...

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